| Pharmaceutical Information |
| Drug Name |
Pentazocine lactate |
| Drug ID |
BADD_D01720 |
| Description |
The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97) |
| Indications and Usage |
For the relief of moderate to severe pain. |
| Marketing Status |
approved; vet_approved |
| ATC Code |
N02AD01 |
| DrugBank ID |
DB00652
|
| KEGG ID |
D02111
|
| MeSH ID |
D010423
|
| PubChem ID |
656697
|
| TTD Drug ID |
D0W6DG
|
| NDC Product Code |
48087-0007 |
| UNII |
1P2XIB510O
|
| Synonyms |
Pentazocine | Lexir | Pentazocine Lactate | Lactate, Pentazocine | Talwin | Fortral | Pentazocine Hydrochloride | Hydrochloride, Pentazocine |
|
| Chemical Information |
| Molecular Formula |
C22H33NO4 |
| CAS Registry Number |
17146-95-1 |
| SMILES |
CC1C2CC3=C(C1(CCN2CC=C(C)C)C)C=C(C=C3)O.CC(C(=O)O)O |
| Chemical Structure |
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| ADRs Induced by Drug |
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